Silver-mediated oxidative C-H difluoromethylation of phenanthridines and 1,10-phenanthrolines.

作者: Sheng-Qing Zhu , Xiu-Hua Xu , Feng-Ling Qing

DOI: 10.1039/C7CC05411D

关键词:

摘要: A silver-mediated oxidative difluoromethylation of phenanthridines and 1,10-phenanthrolines with TMSCF2H is disclosed. This C–H N-containing polycyclic aromatics constitutes an efficient method for the regioselective synthesis difluoromethylated N-heterocycles.

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