Inhibitors of protein tyrosine kinases

作者: David W Fry , Alexander J Bridges

DOI: 10.1016/0958-1669(95)80109-X

关键词:

摘要: The description in the past year of several novel protein tyrosine kinase inhibitors, which exhibit dramatic improvements potency and specificity over earlier agents, will be considered a major turning point field. These compounds appear to have necessary pharmacological properties finally allow clarification whether suppression specific kinases is therapeutic benefit certain disease states.

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