GSK-3-Selective Inhibitors Derived from Tyrian Purple Indirubins
作者： Maryse Leost , Xiaozhou P. Ryan , Claudia Alin Vonica , Ali Brivanlou , Rana Dajani
DOI: 10.1016/J.CHEMBIOL.2003.11.010
关键词:
摘要: … natural product, turned out to be a potent GSK-3 inhibitor. Its synthetic derivative, 6-… inhibitors of GSK-3. We here provide the first cocrystal structures of GSK-3 and CDK5 with an inhibitor…
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