Characterization of potent inhibitors of the Bcr-Abl and the c-kit receptor tyrosine kinases.

作者: John Kuriyan , John Kuriyan , Bayard Clarkson , David Wisniewski , Bhushan Nagar

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摘要: … with imatinib to inhibit Bcr-Abl-… Bcr-Abl resemble those detected during c-kit signal transduction (57), we set out to dissect src family kinase-dependent target phosphorylation in the c-kit …

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