25 years of small molecular weight kinase inhibitors: potentials and limitations.

作者: Doriano Fabbro

DOI: 10.1124/MOL.114.095489

关键词:

摘要: … With a few exceptions, like the rapalogs (everolimus and temsirolimus) and trametinib, all of the small molecular weight kinase inhibitors are directed toward the ATP-binding site. The …

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