β-Sultams exhibit discrete binding preferences for diverse bacterial enzymes with nucleophilic residues
作者： Roman Kolb , Nina C. Bach , Stephan A. Sieber
DOI: 10.1039/C3CC46002A
关键词:
摘要: β-Sultams are potent electrophiles that modify nucleophilic residues in selected enzyme active sites. We here identify and characterize some of the specific bacterial targets show a unique inhibition azoreductase family.
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