A small molecule–kinase interaction map for clinical kinase inhibitors

作者: Miles A Fabian , William H Biggs , Daniel K Treiber , Corey E Atteridge , Mihai D Azimioara

DOI: 10.1038/NBT1068

关键词:

摘要: … of these compounds target the kinase ATP … kinases in addition to their known, primary targets. For most of the compounds tested here, the tightest interaction is with the kinase or kinases …

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