Novel synthesis of the pharmacologically important 1-substituted-6-phenyl-4H-s-triazolo[4,3-a][1,4]benzodiazepines

作者: Jackson B. Hester

DOI: 10.1002/JHET.5570170331

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摘要: Several 6-phenyl-4H-s-triazolo[4,3-a][1,4]benzodiazepines have useful biological activity both in experimental animals and man. This manuscript describes a novel synthesis of these compounds from intermediates that do not pre-formed benzodiazepine ring system.

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