The Current State of Peptide Drug Discovery: Back to the Future?
作者： Antoine Henninot , James C. Collins , John M. Nuss
DOI: 10.1021/ACS.JMEDCHEM.7B00318
关键词:
摘要: … However, elegant new approaches as outlined in section 3.4 have brought insulin … in nature and will provide new targets for peptide discovery, if a lead can be found and optimized. …
acs.org
sci-hub.se 参考文章(289)
Sung In Lim, Inchan Kwon, Bioconjugation of therapeutic proteins and enzymes using the expanded set of genetically encoded amino acids Critical Reviews in Biotechnology. ,vol. 36, pp. 803- 815 ,(2016) , 10.3109/07388551.2015.1048504
Michael Seia, Einat Zisman, Different roles of D-amino acids in immune phenomena. The FASEB Journal. ,vol. 11, pp. 449- 456 ,(1997) , 10.1096/FASEBJ.11.6.9194525
Stanislav I. Presolski, Vu Phong Hong, M.G. Finn, Copper-Catalyzed Azide–Alkyne Click Chemistry for Bioconjugation Current protocols in chemical biology. ,vol. 3, pp. 153- 162 ,(2011) , 10.1002/9780470559277.CH110148
Christopher T. Walsh, Insights into the chemical logic and enzymatic machinery of NRPS assembly lines. Natural Product Reports. ,vol. 33, pp. 127- 135 ,(2016) , 10.1039/C5NP00035A
Chewn-Lang Ho, Yah-Luen Lin, Wan-Chen Chen, Raniero Rocchi, Tom Piek, Comparison of the immunogenicity of wasp venom peptides with or without carbohydrate moieties Toxicon. ,vol. 36, pp. 217- 221 ,(1998) , 10.1016/S0041-0101(97)00066-4
Denise Wootten, Arthur Christopoulos, Patrick M. Sexton, Emerging paradigms in GPCR allostery: implications for drug discovery Nature Reviews Drug Discovery. ,vol. 12, pp. 630- 644 ,(2013) , 10.1038/NRD4052
M. Cristina Castelli, Diane F. Wong, Kristen Friedman, M. Gary I. Riley, Pharmacokinetics of oral cyanocobalamin formulated with sodium N-[8-(2-hydroxybenzoyl)amino]caprylate (SNAC): an open-label, randomized, single-dose, parallel-group study in healthy male subjects. Clinical Therapeutics. ,vol. 33, pp. 934- 945 ,(2011) , 10.1016/J.CLINTHERA.2011.05.088
Yollete V. Guillen Schlippe, Matthew C. T. Hartman, Kristopher Josephson, Jack W. Szostak, In vitro selection of highly modified cyclic peptides that act as tight binding inhibitors. Journal of the American Chemical Society. ,vol. 134, pp. 10469- 10477 ,(2012) , 10.1021/JA301017Y
David W. Wood, Julio A. Camarero, Intein Applications: From Protein Purification and Labeling to Metabolic Control Methods Journal of Biological Chemistry. ,vol. 289, pp. 14512- 14519 ,(2014) , 10.1074/JBC.R114.552653
V. Cardona, I. Eberle, S. Barthélémy, J. Beythien, B. Doerner, P. Schneeberger, J. Keyte, P. D. White, Application of Dmb-Dipeptides in the Fmoc SPPS of Difficult and Aspartimide-Prone Sequences International Journal of Peptide Research and Therapeutics. ,vol. 14, pp. 285- 292 ,(2008) , 10.1007/S10989-008-9154-Z