Triazole-Containing Releasable Linkers, Conjugates Thereof, and Methods of Preparation
作者： Patrick Henry Beusker , Franciscus Marinus Hendrikus De Groot
DOI:
关键词: Combinatorial chemistry 、 Triazole 、 Linker 、 Conjugate 、 Moiety 、 Chemistry
摘要: This invention relates to compounds comprising one or more therapeutic and/or diagnostic moieties and functional linked together via triazole-containing linkers their intermediates methods of preparation. The linker may optionally contain conditionally-cleavable conditionally-transformable spacer systems in between said moiety/moieties the moieties.
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